{"product_id":"acetato-de-trembolona-150mg-ml","title":"Acetato de Trembolona 100mg\/ml","description":"\u003ch2 data-path-to-node=\"1\"\u003eSeção | Descrição Técnica\u003c\/h2\u003e\n\u003cp data-path-to-node=\"2\"\u003e\u003cb data-path-to-node=\"2\" data-index-in-node=\"0\"\u003eNome do produto\u003c\/b\u003e Acetato de Trembolona 100 mg\/mL\u003c\/p\u003e\n\u003cp data-path-to-node=\"3\"\u003e\u003cb data-path-to-node=\"3\" data-index-in-node=\"0\"\u003ePrincípio ativo\u003c\/b\u003e Acetato de Trembolona\u003c\/p\u003e\n\u003cp data-path-to-node=\"4\"\u003e\u003cb data-path-to-node=\"4\" data-index-in-node=\"0\"\u003eCAS\u003c\/b\u003e 10161-34-9\u003c\/p\u003e\n\u003cp data-path-to-node=\"5\"\u003e\u003cb data-path-to-node=\"5\" data-index-in-node=\"0\"\u003eClasse farmacológica\u003c\/b\u003e Andrógeno esteroide anabolizante; éster de liberação rápida\u003c\/p\u003e\n\u003cp data-path-to-node=\"6\"\u003e\u003cb data-path-to-node=\"6\" data-index-in-node=\"0\"\u003eForma farmacêutica\u003c\/b\u003e Solução oleosa estéril para uso parenteral\u003c\/p\u003e\n\u003cp data-path-to-node=\"7\"\u003e\u003cb data-path-to-node=\"7\" data-index-in-node=\"0\"\u003eApresentação\u003c\/b\u003e Frasco-ampola de vidro de 10 mL\u003c\/p\u003e\n\u003cp data-path-to-node=\"8\"\u003e\u003cb data-path-to-node=\"8\" data-index-in-node=\"0\"\u003eConcentração\u003c\/b\u003e 100 mg\/mL\u003c\/p\u003e\n\u003cp data-path-to-node=\"9\"\u003e\u003cb data-path-to-node=\"9\" data-index-in-node=\"0\"\u003eComposição por mL\u003c\/b\u003e * Acetato de Trembolona: 100 mg\u003c\/p\u003e\n\u003cul data-path-to-node=\"10\"\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"10,0,0\"\u003eVeículo oleoso USP (ex: óleo de semente de uva ou óleo MCT): q.s.p. 1 mL\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"10,1,0\"\u003eAntioxidantes e estabilizantes inativos\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp data-path-to-node=\"11\"\u003e\u003cb data-path-to-node=\"11\" data-index-in-node=\"0\"\u003eAparência da solução\u003c\/b\u003e Solução oleosa transparente, cor amarelo claro a âmbar\u003c\/p\u003e\n\u003cp data-path-to-node=\"12\"\u003e\u003cb data-path-to-node=\"12\" data-index-in-node=\"0\"\u003ePropriedades físico-químicas (IFA - Insumo Farmacêutico Ativo)\u003c\/b\u003e * \u003cb data-path-to-node=\"12\" data-index-in-node=\"65\"\u003eAspecto:\u003c\/b\u003e pó cristalino amarelo pálido\u003c\/p\u003e\n\u003cul data-path-to-node=\"13\"\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"13,0,0\"\u003e\u003cb data-path-to-node=\"13,0,0\" data-index-in-node=\"0\"\u003ePonto de fusão:\u003c\/b\u003e 90–93 °C\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"13,1,0\"\u003e\u003cb data-path-to-node=\"13,1,0\" data-index-in-node=\"0\"\u003ePeso molecular:\u003c\/b\u003e 312,41 g\/mol\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"13,2,0\"\u003e\u003cb data-path-to-node=\"13,2,0\" data-index-in-node=\"0\"\u003eSolubilidade:\u003c\/b\u003e insolúvel em água; solúvel em óleos e solventes orgânicos\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp data-path-to-node=\"14\"\u003e\u003cb data-path-to-node=\"14\" data-index-in-node=\"0\"\u003ePropriedades físico-químicas (solução)\u003c\/b\u003e * \u003cb data-path-to-node=\"14\" data-index-in-node=\"41\"\u003eDensidade:\u003c\/b\u003e 0,90–0,94 g\/mL (25 °C)\u003c\/p\u003e\n\u003cul data-path-to-node=\"15\"\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"15,0,0\"\u003e\u003cb data-path-to-node=\"15,0,0\" data-index-in-node=\"0\"\u003eViscosidade:\u003c\/b\u003e moderada\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"15,1,0\"\u003e\u003cb data-path-to-node=\"15,1,0\" data-index-in-node=\"0\"\u003epH:\u003c\/b\u003e não aplicável (solução não aquosa)\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp data-path-to-node=\"16\"\u003e\u003cb data-path-to-node=\"16\" data-index-in-node=\"0\"\u003eEsterilidade\u003c\/b\u003e Cumpre USP \u0026lt;71\u0026gt;\u003c\/p\u003e\n\u003cp data-path-to-node=\"17\"\u003e\u003cb data-path-to-node=\"17\" data-index-in-node=\"0\"\u003eFarmacodinâmica\u003c\/b\u003e Potente agonista dos receptores androgênicos. Não aromatiza em estrogênios. Apresenta alta atividade anabólica e androgênica, com forte afinidade pelo receptor androgênico. O éster acetato permite uma liberação rápida a partir do local de administração.\u003c\/p\u003e\n\u003cp data-path-to-node=\"18\"\u003e\u003cb data-path-to-node=\"18\" data-index-in-node=\"0\"\u003eFarmacocinética\u003c\/b\u003e * \u003cb data-path-to-node=\"18\" data-index-in-node=\"18\"\u003eAbsorção:\u003c\/b\u003e Rápida absorção a partir do depósito oleoso intramuscular.\u003c\/p\u003e\n\u003cul data-path-to-node=\"19\"\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"19,0,0\"\u003e\u003cb data-path-to-node=\"19,0,0\" data-index-in-node=\"0\"\u003eDistribuição:\u003c\/b\u003e Alta afinidade por tecidos ricos em receptores androgênicos; ligação moderada a proteínas plasmáticas.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"19,1,0\"\u003e\u003cb data-path-to-node=\"19,1,0\" data-index-in-node=\"0\"\u003eMetabolismo:\u003c\/b\u003e Metabolização hepática mediante redução e conjugação; não sofre aromatização.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"19,2,0\"\u003e\u003cb data-path-to-node=\"19,2,0\" data-index-in-node=\"0\"\u003eEliminação:\u003c\/b\u003e Principalmente renal na forma de metabólitos conjugados; pequena fração fecal.\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"19,3,0\"\u003e\u003cb data-path-to-node=\"19,3,0\" data-index-in-node=\"0\"\u003eMeia-vida:\u003c\/b\u003e Aproximadamente 2–3 dias\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp data-path-to-node=\"20\"\u003e\u003cb data-path-to-node=\"20\" data-index-in-node=\"0\"\u003eEstabilidade\u003c\/b\u003e Sensível à luz e à oxidação; estável sob condições adequadas de armazenamento.\u003c\/p\u003e\n\u003cp data-path-to-node=\"21\"\u003e\u003cb data-path-to-node=\"21\" data-index-in-node=\"0\"\u003eControles de qualidade típicos\u003c\/b\u003e * Pureza ≥ 97–99%\u003c\/p\u003e\n\u003cul data-path-to-node=\"22\"\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"22,0,0\"\u003eIdentificação do IFA por HPLC\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"22,1,0\"\u003eEnsaio de teor\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"22,2,0\"\u003eImpurezas relacionadas\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp data-path-to-node=\"22,3,0\"\u003eTestes de esterilidade e endotoxinas bacterianas\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp data-path-to-node=\"23\"\u003e\u003cb data-path-to-node=\"23\" data-index-in-node=\"0\"\u003eCondições de conservação\u003c\/b\u003e Conservar entre 15–25 °C; proteger da luz; não congelar; manter na embalagem original hermeticamente fechada.\u003c\/p\u003e\n\u003cp data-path-to-node=\"24\"\u003e\u003cb data-path-to-node=\"24\" data-index-in-node=\"0\"\u003eRestrições legais\u003c\/b\u003e Substância controlada em múltiplas jurisdições. Uso restrito e sujeito à regulamentação sanitária; apenas sob prescrição e supervisão profissional, conforme a legislação local.\u003c\/p\u003e\n\u003ch3 data-start=\"170\" data-end=\"203\"\u003e\n\u003cbr\u003e\u003cbr\u003e\n\u003c\/h3\u003e","brand":"Wallgen Labs","offers":[{"title":"Default Title","offer_id":52208213852465,"sku":null,"price":360.0,"currency_code":"BRL","in_stock":false}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0966\/0497\/9505\/files\/Acetatodetrembo.png?v=1765840727","url":"https:\/\/wellgenlabs.org\/products\/acetato-de-trembolona-150mg-ml","provider":"Wellgen Labs","version":"1.0","type":"link"}